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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T14895 | Tanzisertib | CC-930 | JNK |
Tanzisertib (CC-930) (CC-930) is a potent inhibitor of JNK1/2/3 with IC50s of 61/7/6 nM, respectively, with potential antifibrotic activity. | |||
T28501 | Ragaglitazar | NNC61-0029,NN-622,(-)-DRF-2725,NNC-61-0029,NN 622,NNC 61-0029 | PPAR |
Ragaglitazar(NNC-61-0029) is a potent dual PPARα and PPARγ agonist that has shown potent lipid-lowering and insulin sensitizing effects in animal models.Ragaglitazar can be used to study type 2 diabetes. | |||
T6776 | BAY 61-3606 dihydrochloride | BAY 61-3606,BAY-61-3606 dihydrochloride | Apoptosis , Syk |
BAY 61-3606 dihydrochloride (BAY 61-3606) is a potent and selective inhibitor of Syk kinase (Ki = 7.5 nM). | |||
T17243 | VU0463271 | N-Cyclopropyl-N-(4-methyl-2-thiazolyl)-2-[(6-phenyl-3-pyridazinyl)thio]acetamide | Potassium Channel |
VU0463271 (N-Cyclopropyl-N-(4-methyl-2-thiazolyl)-2-[(6-phenyl-3-pyridazinyl)thio]acetamide) is a potent and selective antagonist of the neuronal-specific potassium-chloride cotransporter 2 (KCC2), with an IC50 of 61 nM ... | |||
T9100 | BP 897 | 2-Naphthalenecarboxamide, N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]- | Dopamine Receptor |
BP 897 (2-Naphthalenecarboxamide, N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]-) is a potent and selective dopamine D3 receptor agonist, and a weak dopamine D2 receptor antagonist, with Kis of 0.92 nM and 61 nM for D3 ... | |||
T1839 | Mps1-IN-2 | Kinesin , PLK | |
Mps1-IN-2 is a potent, selective and ATP-competitive dual Mps1/Plk1 inhibitor. | |||
T4263 | BAY 61-3606 | Syk inhibitor IV | Apoptosis , Syk |
BAY 61-3606 (Syk inhibitor IV) is a potent, ATP-competitive, reversible, and highly selective inhibitor of Syk tyrosine kinase activity (Ki= 7.5 nM), exhibiting no inhibitory effect against Btk, Fyn, Itk, Lyn, and Src. | |||
T38238 | 2'-Deoxy-2'-fluorocytidine | Nucleoside Antimetabolite/Analog , Influenza Virus | |
2'-Deoxy-2'-fluorocytidine, an nucleoside analog, is a potent inhibitor of Crimean-Congo hemorrhagic fever virus (CCHFV) replication. 2′-deoxy-2′-fluorocytidine can act synergistically with T705 to increase the potency o... | |||
T69545 | Mpro 61 | ||
Mpro 61 is a potent non-covalent inhibitor of SARS-CoV-2 main protease. | |||
T76284 | β-Lipotropin (61-69) | ||
β-Lipotropin (61-69) is a potent opioid agonist [1] [2] . | |||
T79426 | SARS-CoV-2-IN-61 | SARS-CoV | |
SARS-CoV-2-IN-61 (compound 8i) is a potent inhibitor of the SARS-CoV-2 PLpro, exhibiting an IC50 of 16 µM and demonstrating antiviral activities [1]. | |||
T65585 | Gefitinib impurity 5 | ||
Gefitinib impurity 5 is a useful organic compound for research related to life sciences. The catalog number is T65585 and the CAS number is 199327-61-2. | |||
T9313 | Imidazopyridine 2 | ||
imidazopyridine 2 is a useful organic compound for research related to life sciences. The catalog number is T9313 and the CAS number is 1256032-61-7. | |||
TN5806 | Ethyl β-D-apiofuranoside | ||
Ethyl β-D-apiofuranoside is a natural product for research related to life sciences. The catalog number is TN5806 and the CAS number is 1932405-61-2. | |||
T61315 | HDAC6/HSP90-IN-2 | ||
HDAC6/HSP90-IN-2 (compound 6e) is a dual inhibitor targeting HDAC6 and Hsp90, exhibiting IC50 values of 105.7 nM and 61 nM, respectively. It is primarily utilized in cancer research [1]. | |||
TN3980 | Epoxyparvinolide | Others | |
Epoxyparvinolide is a natural product of Pogostemon, Lamiaceae. The catalog number is TN3980 and the CAS number is 102227-61-2. Epoxyparvinolide can be used as a reference standard. | |||
T60381 | LSD1-IN-12 | ||
LSD1-IN-12 (compound 2) is an effective inhibitor of LSD1, demonstrating inhibitory Ki values of 1.1 μM (LSD1), 61 μM (LSD2), 2.3 μM (MAO-A), and 3.5 μM (MAO-B), respectively [1]. | |||
T76199 | α-Synuclein (61-75) (TFA) | ||
α-Synuclein (61-75) TFA is a fragment (residues 61-75) of the abundant neuronal protein α-Synuclein, which is predominantly located in presynaptic nerve terminals. α-Synuclein serves as a potential biomarker for Parkinso... | |||
T126388 | 9-Oxotournefortiolide, Tourneforin | ||
9-Oxotournefortiolide, Tourneforin is a useful organic compound for research related to life sciences. The catalog number is T126388 and the CAS number is 111420-61-2. | |||
T64444 | 2-Hydroxy-N-phenylacetamide | ||
2-Hydroxy-N-phenylacetamide is a useful organic compound for research related to life sciences. The catalog number is T64444 and the CAS number is 4746-61-6. |